Journal of enzyme inhibition and medicinal chemistry

369 articles found in (213msec)
Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors.
Marastoni, Mauro Trapella, Claudio Scotti, Alessandra Fantinati, Anna Ferretti, Valeria Marzola, Erika Eleonora, Gallerani Gavioli, Riccardo Preti, Delia
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(32), issue(1),  Dec.2017
Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors.
Ramya, P V Sri Angapelly, Srinivas Angeli, Andrea Digwal, Chander Singh Arifuddin, Mohammed Babu, Bathini Nagendra Supuran, Claudiu T Kamal, Ahmed
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(32), issue(1),  Dec.2017
Bulge oligonucleotide as an inhibitory agent of bacterial topoisomerase I.
Yang, Zhaoqi Jiang, Tuoyu Zhong, Hanshi Kang, Yu
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(33), issue(1),  Dec.2018
Cholesterol sulfate as a potential inhibitor of hepatitis C virus NS3 helicase.
Furuta, Atsushi Salam, Kazi Abdus Akimitsu, Nobuyoshi Tanaka, Junichi Tani, Hidenori Yamashita, Atsuya Moriishi, Kohji Nakakoshi, Masamichi Tsubuki, Masayoshi Sekiguchi, Yuji Tsuneda, Satoshi Noda, Naohiro
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(29), issue(2),  Apr.2014
Sulfonamide-metal complexes endowed with potent anti-Trypanosoma cruzi activity.
Chohan, Zahid H Hernandes, Marcelo Zaldini Sensato, Fabricio R Moreira, Diogo Rodrigo Magalhaes Pereira, Valéria Rego Alves Neves, Juliana Kelle de Andrade Lemoine de Oliveira, Andresa Pereira de Oliveira, Beatriz Coutinho Leite, Ana Cristina Lima
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(29), issue(2),  Apr.2014
More effective dithiocarbamate derivatives inhibiting carbonic anhydrases, generated by QSAR and computational design.
Avram, Speranta Milac, Adina Luminita Carta, Fabrizio Supuran, Claudiu T
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(28), issue(2),  Apr.2013
In vitro antibacterial, antifungal and cytotoxic activities of some triazole Schiff bases and their oxovanadium(IV) complexes.
Sumrra, Sajjad H Chohan, Zahid H
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(28), issue(6),  Dec.2013
Effects of novel human cathepsin S inhibitors on cell migration in human cancer cells.
Tsai, Ju-Ying Lee, Mon-Juan Chang, Margaret Dah-Tsyr Wang, Hsin-Chieh Lin, Chun-Cheng Huang, Haimei
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(29), issue(4),  Aug.2014
Monoclonal antibodies raised against 167-180 aa sequence of human carbonic anhydrase XII inhibit its enzymatic activity.
Dekaminaviciute, Dovile Kairys, Visvaldas Zilnyte, Milda Petrikaite, Vilma Jogaite, Vaida Matuliene, Jurgita Gudleviciene, Zivile Vullo, Daniela Supuran, Claudiu T Zvirbliene, Aurelija
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(29), issue(6),  Dec.2014
Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel cyanoenone and enone benzenesulfonamides.
Ghorab, Mostafa M Higgins, Maureen Alsaid, Mansour S Arafa, Reem K Shahat, Abdelaaty A Dinkova-Kostova, Albena T
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(29), issue(6),  Dec.2014
Citrus medica L. cv Diamante (Rutaceae) peel extract improves glycaemic status of Zucker diabetic fatty (ZDF) rats and protects against oxidative stress.
Menichini, Francesco Tundis, Rosa Loizzo, Monica R Bonesi, Marco D'Angelo, Danila Lombardi, Pietro Mastellone, Vincenzo
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(31), issue(6),  Dec.2016
A nonmainstream approach against cancer.
Fais, Stefano
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(31), issue(6),  Dec.2016
Discovery of Strecker-type ?-aminonitriles as a new class of human carbonic anhydrase inhibitors using differential scanning fluorimetry.
Krasavin, Mikhail Stavniichuk, Roman Zozulya, Sergey Borysko, Petro Vullo, Daniela Supuran, Claudiu T
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(31), issue(6),  Dec.2016
Effects of prodigiosin family compounds from Pseudoalteromonas sp. 1020R on the activities of protein phosphatases and protein kinases.
Soliev, Azamjon B Hosokawa, Kakushi Enomoto, Keiichi
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(30), issue(4),  
Purification and characterization of a phenoloxidase in the hemocytes of Ephestia kuehniella Zeller (Lepidoptera: Pyralidae): effects of insect growth regulators and endogenous inhibitors.
Delkash-Roudsari, Sahar Zibaee, Arash Bigham, Zargham
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(30), issue(4),  
A new affinity method for purification of bovine testicular hyaluronidase enzyme and an investigation of the effects of some compounds on this enzyme.
Kaya, Mustafa Oguzhan Arslan, Oktay Guler, Ozen Ozensoy
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(30), issue(4),  
Stability and binding effects of silver(I) complexes at lipoxygenase-1.
Vrontaki, Eleni Leonis, Georgios Avramopoulos, Aggelos Papadopoulos, Manthos G Sim?i?, Mihael Grdadolnik, Simona Goli? Afantitis, Antreas Melagraki, Georgia Hadjikakou, Sotiris K Mavromoustakos, Thomas
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(30), issue(4),  
Biological activity of pyrazole and imidazole-dehydroepiandrosterone derivatives on the activity of 17?-hydroxysteroid dehydrogenase.
Cabeza, Marisa Posada, Alejandro Sánchez-Márquez, Araceli Heuze, Yvonne Moreno, Isabel Soriano, Juan Garrido, Mariana Cortés, Francisco Bratoeff, Eugene
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(31), issue(1),  
Evaluation of the anticancer potential of a sulphonamide carbonic anhydrase IX inhibitor on cervical cancer cells.
Koyuncu, Ismail Tülüce, Yasin Slahaddin Qadir, Hewa Durgun, Mustafa Supuran, Claudiu T
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(34), issue(1),  Dec.2019
Identification of cisplatin-binding sites on the large cytoplasmic loop of the Na+/K+-ATPase.
?eflová, Jaroslava ?echová, Petra ?tenclová, Tereza ?ebela, Marek Kubala, Martin
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(33), issue(1),  Dec.2018
Syntheses and evaluation of multicaulin and miltirone-like compounds as antituberculosis agents.
Burmao?lu, Serdar Seçinti, Hatice Mozio?lu, Erkan Gören, Ahmet C Altunda?, Ramazan Seçen, Hasan
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(32), issue(1),  Dec.2017
Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A receptor.
Duroux, Romain Renault, Nicolas Cuelho, Joana Esteves Agouridas, Laurence Blum, David Lopes, Luisa V Melnyk, Patricia Yous, Saďd
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(32), issue(1),  Dec.2017
Nitroimidazole-based inhibitors DTP338 and DTP348 are safe for zebrafish embryos and efficiently inhibit the activity of human CA IX in Xenopus oocytes.
Aspatwar, Ashok Becker, Holger M Parvathaneni, Nanda Kumar Hammaren, Milka Svorjova, Aleksandra Barker, Harlan Supuran, Claudiu T Dubois, Ludwig Lambin, Philippe Parikka, Mataleena Parkkila, Seppo Winum, Jean-Yves
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(33), issue(1),  Dec.2018
Synthesis and biological evaluation of dithiocarbamate esters of parthenolide as potential anti-acute myelogenous leukaemia agents.
Ding, Yahui Yang, Zhongjin Ge, Weizhi Kuang, Beijia Xu, Junqing Yang, Juan Chen, Yue Zhang, Quan
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(33), issue(1),  Dec.2018
Reliability analysis and optimization of the consensus docking approach for the development of virtual screening studies.
Poli, Giulio Martinelli, Adriano Tuccinardi, Tiziano
Journal of enzyme inhibition and medicinal chemistry (J Enzyme Inhib Med Chem),vol(31), issue(sup2),  

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